瑞卡帕布樟脑磺酸盐 Rucaparib Camsylate 是 PARP 的抑制剂,对PARP1的 Ki 值为1.4 nM。也可结合PARP其他八个结构域。
中文别名:
英文同义词: RUCAPARIB CAMSYLATE; 芦卡帕利; 8‐Fluoro‐2‐(4‐methylaminomethyl‐phenyl)‐1,3,4,5‐tetrahydro‐azepino[5,4,3‐cd] indol‐6‐one (S)‐camphorsulfonate Salt;
英文名称:
[4-(8-fluoro-6-oxo-3,4,5,6-tetrahydro-1h-azepino[5,4,3-cd]indol-2-yl)phenyl]-n-methylmethanaminium [(1s,4r)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonate; rucaparib camsylate; CHEBI:134692; co-338;